CAS 540769-28-6: Palosuran

CAS 540769-28-6: Palosuran
(World's Largest Pharmaceutical Supplier)

  • CAS Number: 540769-28-6
  • Stock: 268g
  • Assay: 99.20%

Palosuran, CAS 540769-28-6

Palosuran, CAS 540769-28-6, Stock 268g, Assay 99.20%, Off-white or White powder, EOS Med Chem is big manufacturer of Palosuran.


Palosuran

Palosuran, also known as ACT-058362, is a Urotensin-II receptor antagonist. Urotensin inhibition with palosuran could be a promising alternative in pulmonary arterial hypertension. Palosuran inhibits binding to primate UT receptors in cell membranes but demonstrates differential activity in intact cells and vascular tissues. Palosuran improves pancreatic and renal function in diabetic rats.


Product Details:

Name: Palosuran

CAS#: 540769-28-6

Chemical Formula: C25H30N4O2

Exact Mass: 418.2369

Molecular Weight: 418.541

Elemental Analysis: C, 71.74; H, 7.23; N, 13.39; O, 7.65


Specification:

Synonym: Palosuran; ACT-058362; ACT058362; ACT 058362.

IUPAC/Chemical Name: 1-(2-(4-benzyl-4-hydroxypiperidin-1-yl)ethyl)-3-(2-methylquinolin-4-yl)urea

InChi Key: WYJCYXOCHXWTHG-UHFFFAOYSA-N

InChi Code: InChI=1S/C25H30N4O2/c1-19-17-23(21-9-5-6-10-22(21)27-19)28-24(30)26-13-16-29-14-11-25(31,12-15-29)18-20-7-3-2-4-8-20/h2-10,17,31H,11-16,18H2,1H3,(H2,26,27,28,30)

SMILES Code: O=C(NC1=CC(C)=NC2=CC=CC=C12)NCCN3CCC(CC4=CC=CC=C4)(O)CC3

Appearance: Solid powder

Purity: >99% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: Soluble in DMSO

Shelf Life: >2 years if stored properly

Drug Formulation: This drug may be formulated in DMSO

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001


Certifications: