CAS 1001389-72-5 : GSK1482160
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GSK1482160, CAS 1001389-72-5

GSK1482160, CAS 1001389-72-5, Stock 343g, Assay 99.29%, White powder, Water 0.38%, Single Impurity 0.33%.

GSK1482160

GSK1482160 is a potent and selective P2X7 receptor allosteric modulator with nanomolar binding affinity and high selectivity. GSK1482160 has been successfully radiolabeled and utilized for imaging P2X7 levels in a mouse model of lipopolysaccharide-induced systemic inflammation.

Product Details:

Name: GSK1482160

CAS#: 1001389-72-5

Chemical Formula: C14H14ClF3N2O2

Exact Mass: 334.0696

Molecular Weight: 334.7232

Elemental Analysis: C, 50.24; H, 4.22; Cl, 10.59; F, 17.03; N, 8.37; O, 9.56

Specification:

Synonym: GSK1482160; GSK-1482160; GSK 1482160.

IUPAC/Chemical Name: (2S)-N-[[2-Chloro-3-(trifluoromethyl)phenyl]methyl]-1-methyl-5-oxo-2-pyrrolidinecarboxamide

InChi Key: IHRKNQDNYKZPNL-JTQLQIEISA-N

InChi Code: InChI=1S/C14H14ClF3N2O2/c1-20(13(22)10-5-6-11(21)19-10)7-8-3-2-4-9(12(8)15)14(16,17)18/h2-4,10H,5-7H2,1H3,(H,19,21)/t10-/m0/s1

SMILES Code: ClC1=C(C=CC=C1CN(C([C@@H]2CCC(N2)=O)=O)C)C(F)(F)F

Appearance: Solid powder

Purity: >99% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: Soluble in DMSO

Shelf Life: >2 years if stored properly

Drug Formulation: This drug may be formulated in DMSO

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001

Certifications: