Gepirone, CAS 83928-76-1

Gepirone, CAS 83928-76-1, Stock 179g, Assay 98.35%, White powder, Water 0.12%, Single Impurity 0.19%.

Gepirone

 Gepirone is a selective 5-HT(1A) agonist that significantly reduces depression. Gepirone is a drug of the azapirone group which is a 5-HT1A receptor agonist belonging to the buspirone family. Gepirone has been shown to be more effective than selective serotonin reuptake inhibitors (SSRIs), as this drug treats the psychiatric disorders without causing sexual dysfunction, which limits the use of SSRIs. It possesses greater selectivity for the 5-HT1A receptor than SSRIs. Clinical studies have shown that gepirone has differential action at pre- and postsynaptic 5-HT1A receptors.

Product Details:

Name: Gepirone

CAS#: 83928-76-1 (free base)

Chemical Formula: C19H29N5O2

Exact Mass: 359.23

Molecular Weight: 359.474

Elemental Analysis: C, 63.48; H, 8.13; N, 19.48; O, 8.90

Specification:

Synonym: Lirafugratinib; RLY-4008; RLY 4008; RLY4008;

IUPAC/Chemical Name: N-[4-(4-amino-5-{3-fluoro-4-[(4-methylpyrimidin-2-yl)oxy]phenyl}-7-methyl-7H-pyrrolo[2,3-d]pyrimidin-6-yl)phenyl]-2-methylprop-2-enamide

InChi Key: XOQVZSSDIQQUGO-UHFFFAOYSA-N

InChi Code: InChI=1S/C28H24FN7O2/c1-15(2)27(37)35-19-8-5-17(6-9-19)24-22(23-25(30)32-14-33-26(23)36(24)4)18-7-10-21(20(29)13-18)38-28-31-12-11-16(3)34-28/h5-14H,1H2,2-4H3,(H,35,37)(H2,30,32,33)

SMILES Code: C=C(C)C(NC1=CC=C(C2=C(C3=CC=C(OC4=NC=CC(C)=N4)C(F)=C3)C5=C(N)N=CN=C5N2C)C=C1)=O

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Shelf Life: >2 years if stored properly

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001